Pharos : Ligand Details - GH396M1YM2XH

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: (1S,9aR,11aS)-9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid phenylamide

PubChem: 44275381

ChEMBL: CHEMBL280155

LyCHI: GH396M1YM2XH

Target Activities

SRD5A1

Tclin

3-oxo-5-alpha-steroid 4-dehydrogenase 1

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.62		J. Med. Chem., (1995) 38:14:2621	7629802

Ki	6.62		J. Med. Chem., (1997) 40:9:1293	9135028

SRD5A2

Tclin

3-oxo-5-alpha-steroid 4-dehydrogenase 2

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.85		J. Med. Chem., (1997) 40:9:1293	9135028

IC50	8.85		J. Med. Chem., (1995) 38:14:2621	7629802

HSD3B1

Tchem

3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	8		J. Med. Chem., (1997) 40:9:1293	9135028