SID103904192
Ligand Summary
Target Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
CDK1
Cyclin-dependent kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
CDK2
Cyclin-dependent kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
CSNK1G1
Casein kinase I isoform gamma-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
CSNK1G2
Casein kinase I isoform gamma-2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
JAK3
Tyrosine-protein kinase JAK3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
ROCK1
Rho-associated protein kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
PRKCD
Protein kinase C delta type
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
CDK7
Cyclin-dependent kinase 7
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
PRKACA
cAMP-dependent protein kinase catalytic subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
SLK
STE20-like serine/threonine-protein kinase
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
RPS6KA5
Ribosomal protein S6 kinase alpha-5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
CDC42BPA
Serine/threonine-protein kinase MRCK alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
CSNK1G3
Casein kinase I isoform gamma-3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
PKN2
Serine/threonine-protein kinase N2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
PRKAA1
5'-AMP-activated protein kinase catalytic subunit alpha-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
ROCK2
Rho-associated protein kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
CDK5
Cyclin-dependent-like kinase 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||