US9206139, 2
Ligand Summary
Target Activities
ADAMTS5
A disintegrin and metalloproteinase with thrombospondin motifs 5
3 Activities
ADAMTS4
A disintegrin and metalloproteinase with thrombospondin motifs 4
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.7 | None, (2015) None:None:None | ||||
IC50 | 8.7 | J Med Chem, (2017) 60:13:5933 | ||||
MMP12
Macrophage metalloelastase
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.58 | None, (2015) None:None:None | ||||
IC50 | 7.58 | J Med Chem, (2017) 60:13:5933 | ||||
MMP2
72 kDa type IV collagenase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.15 | None, (2015) None:None:None | ||||
MMP9
Matrix metalloproteinase-9
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.36 | None, (2015) None:None:None | ||||
MMP1
Interstitial collagenase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.05 | None, (2015) None:None:None | ||||