Florbetapir F-18
a PET agent for Abeta plaques
Ligand Summary
UNII: 6W15Z5R0RU
PubChem: 24822371
ChEMBL: CHEMBL1774461
DrugCentral: 4285
LyCHI: QN2675BNDU23
Target Activities
APP
Amyloid-beta A4 protein
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.54 | J. Med. Chem., (2010) 53:3:933 | ||||
Ki | 8.54 | ACS Med. Chem. Lett., (2011) 2:9:673 | ||||
Ki | 8.54 | J. Med. Chem., (2011) 54:23:8085 | ||||
Ki | 8.54 | ACS Med. Chem. Lett., (2012) 3:4:265 | ||||
Ki | 8.54 | J. Med. Chem., (2012) 55:2:883 | ||||
Ki | 8.54 | Bioorg. Med. Chem., (2013) 21:13:3708 | ||||
Ki | 8.54 | |||||