CHEMBL432713
Ligand Summary
Name: (E)-3-(3,4-Dichloro-phenyl)-N-{5-[4-(5-hydroxy-1H-indol-3-yl)-piperidin-1-yl]-pentyl}-acrylamide
PubChem: 10436045
Guide to Pharmacology: 782
ChEMBL: CHEMBL432713
LyCHI: FQLZHFYTFTAU
Target Activities
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CCR2
C-C chemokine receptor type 2
8 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
Ki | 7.3 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2006) 16:14:3735 | ||||
Ki | 7.78 | J. Med. Chem., (2003) 46:19:4070 | ||||
7 | ||||||
HTR2C
5-hydroxytryptamine receptor 2C
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.1 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR6
5-hydroxytryptamine receptor 6
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.1 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR7
5-hydroxytryptamine receptor 7
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.2 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1A
5-hydroxytryptamine receptor 1A
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1E
5-hydroxytryptamine receptor 1E
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.2 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1F
5-hydroxytryptamine receptor 1F
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.5 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1B
5-hydroxytryptamine receptor 1B
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.9 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR2A
5-hydroxytryptamine receptor 2A
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.7 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
DRD2
D(2) dopamine receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.8 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||