SB-282241
Ligand Summary
Name: SB-282241
PubChem: 10436045
Guide to Pharmacology: 782
ChEMBL: CHEMBL432713
LyCHI: FQLZHFYTFTAU
Target Activities
CCR2
C-C chemokine receptor type 2
11 Activities
Items per page:
1 – 10 of 11
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
7 | ||||||
Ki | 7.78 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2000) 10:16:1803 | ||||
Ki | 7.3 | J. Med. Chem., (2003) 46:19:4070 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2006) 16:14:3735 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2008) 18:4:1450 | ||||
Ki | 7.3 | Bioorg. Med. Chem. Lett., (2008) 18:4:1450 | ||||
HTR1F
5-hydroxytryptamine receptor 1F
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.5 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
DRD2
D(2) dopamine receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.8 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR2B
5-hydroxytryptamine receptor 2B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.6 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
DRD3
D(3) dopamine receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.1 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1B
5-hydroxytryptamine receptor 1B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.9 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1A
5-hydroxytryptamine receptor 1A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR2A
5-hydroxytryptamine receptor 2A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.7 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR2C
5-hydroxytryptamine receptor 2C
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.1 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR1E
5-hydroxytryptamine receptor 1E
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.2 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR7
5-hydroxytryptamine receptor 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.2 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||
HTR6
5-hydroxytryptamine receptor 6
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 7.1 | Bioorg. Med. Chem. Lett., (2001) 11:16:2177 | ||||