CHEMBL538632
Ligand Summary
Name: 3-(3-(tert-butylthio)-5-(pyridin-2-ylmethoxy)-1-(4-(pyridin-3-yl)benzyl)-1H-indol-2-yl)-2,2-dimethylpropanoic acid
PubChem: 16223851
ChEMBL: CHEMBL538632
LyCHI: FA7ULCQ6NF73
Target Activities
CYP3A4
Cytochrome P450 3A4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.33 | J. Med. Chem., (2009) 52:19:5803 | ||||
CYP2C9
Cytochrome P450 2C9
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.81 | J. Med. Chem., (2009) 52:19:5803 | ||||
ALOX5AP
Arachidonate 5-lipoxygenase-activating protein
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.05 | J. Med. Chem., (2009) 52:19:5803 | ||||
CYP2D6
Cytochrome P450 2D6
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.59 | J. Med. Chem., (2009) 52:19:5803 | ||||