CHEMBL4634092
Ligand Summary
Name: 3-((7-(5-Chloro-3-methyl-2-(((R)-morpholin-2-yl)methyl)phenyl)thieno[3,2-b]pyridin-2-yl)methyl)-3-azabicyclo[3.1.0]hexane-2,4-dione
ChEMBL: CHEMBL4634092
LyCHI: F4M2GZUR26RJ
Target Activities
USP7
Ubiquitin carboxyl-terminal hydrolase 7
2 Activities
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.1 | J Med Chem, (2020) 63:10:5398 | ||||