Pharos : Ligand Details - DXZHCK45G1NL

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: Cenicriviroc

PubChem: 11285791

PubChem: 11285792

ChEMBL: CHEMBL2105686

ChEMBL: CHEMBL2110727

LyCHI: DXZHCK45G1NL

Target Activities

Explore Associated and Predicted Targets

CCR5

Tclin

C-C chemokine receptor type 5

4 Activities

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1 – 4 of 4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	10		J. Med. Chem., (2006) 49:6:2037	16539392

IC50	9.7		J. Med. Chem., (2006) 49:6:2037	16539392

IC50	8.52		J. Med. Chem., (2012) 55:22:9363	22931505

IC50	8.51		J. Med. Chem., (2006) 49:6:2037	16539392

CCR2

Tchem

C-C chemokine receptor type 2

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.23		J. Med. Chem., (2006) 49:6:2037	16539392

IC50	8.23		J. Med. Chem., (2012) 55:22:9363	22931505

IC50	8.23		J Med Chem, (2020) 63:10:5031	31930920

CCR7

Tchem

C-C chemokine receptor type 7

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.51		J Med Chem, (2020) 63:10:5031	31930920