Cenicriviroc
Ligand Summary
Name: Cenicriviroc
PubChem: 11285791
PubChem: 11285792
ChEMBL: CHEMBL2105686
ChEMBL: CHEMBL2110727
LyCHI: DXZHCK45G1NL
Target Activities
CCR5
C-C chemokine receptor type 5
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 10 | J. Med. Chem., (2006) 49:6:2037 | ||||
IC50 | 9.7 | J. Med. Chem., (2006) 49:6:2037 | ||||
IC50 | 8.52 | J. Med. Chem., (2012) 55:22:9363 | ||||
IC50 | 8.51 | J. Med. Chem., (2006) 49:6:2037 | ||||
CCR2
C-C chemokine receptor type 2
3 Activities
CCR7
C-C chemokine receptor type 7
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.51 | J Med Chem, (2020) 63:10:5031 | ||||