CHEMBL2419697
Ligand Summary
Name: CHEMBL2419697::US9181266, 1
PubChem: 136237302
ChEMBL: CHEMBL2419697
LyCHI: DRK86DP8XAP2
Target Activities
TNKS2
Tankyrase-2
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.64 | J. Med. Chem., (2013) 56:16:6495 | ||||
IC50 | 7.64 | None, (2015) None:None:None | ||||
WNT3A
Protein Wnt-3a
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.4 | J. Med. Chem., (2013) 56:16:6495 | ||||
TNKS
Tankyrase-1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.19 | None, (2015) None:None:None | ||||