GI254023X
Ligand Summary
Name: GI254023X
PubChem: 9952396
Guide to Pharmacology: 9687
ChEMBL: CHEMBL1229516
LyCHI: DQ5BF6VS84WR
Target Activities
ADAM10
Disintegrin and metalloproteinase domain-containing protein 10
2 Activities
ADAM17
Disintegrin and metalloproteinase domain-containing protein 17
2 Activities
MMP14
Matrix metalloproteinase-14
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.06 | Eur. J. Med. Chem., (2016) 111:None:193 | ||||
MMP2
72 kDa type IV collagenase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.68 | Eur. J. Med. Chem., (2016) 111:None:193 | ||||
MMP9
Matrix metalloproteinase-9
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.29 | Eur. J. Med. Chem., (2016) 111:None:193 | ||||
MMP1
Interstitial collagenase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.9 | Eur. J. Med. Chem., (2016) 111:None:193 | ||||