CHEMBL3600918
Ligand Summary
Name: (3S,6S,9R,12S,15S,23S)-12-((1H-imidazol-5-yl)methyl)-3-((1H-indol-3-yl)methyl)-15-((R)-2-acetamidohexanamido)-6-(3-guanidinopropyl)-1,7,13-trimethyl-9-(naphthalen-2-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexaazacyclotricosane-23-carboxamide
PubChem: 122184637
ChEMBL: CHEMBL3600918
LyCHI: D6114QQVTB1J
Target Activities
MC1R
Melanocyte-stimulating hormone receptor
2 Activities
MC4R
Melanocortin receptor 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.4 | J. Med. Chem., (2015) 58:16:6359 | ||||
MC3R
Melanocortin receptor 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.6 | J. Med. Chem., (2015) 58:16:6359 | ||||
MC5R
Melanocortin receptor 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.55 | J. Med. Chem., (2015) 58:16:6359 | ||||