Pharos : Ligand Details - D5LDVLDUNMFY

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: linopirdine

PubChem: 3932

Guide to Pharmacology: 2599

ChEMBL: CHEMBL319111

LyCHI: D5LDVLDUNMFY

Target Activities

Explore Associated and Predicted Targets

KCNQ1

Tclin

Potassium voltage-gated channel subfamily KQT member 1

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	4.4			12690036

KCNQ2

Tclin

Potassium voltage-gated channel subfamily KQT member 2

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	5.3			9836639

KCNQ3

Tclin

Potassium voltage-gated channel subfamily KQT member 3

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	5.4			9836639

KCNQ4

Tclin

Potassium voltage-gated channel subfamily KQT member 4

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	4.9			11245603

KCNQ5

Tclin

Potassium voltage-gated channel subfamily KQT member 5

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	4.8			10787416

CYP3A4

Tclin

Cytochrome P450 3A4

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
AC50	6.3		None, None:None:None

CYP2C19

Tchem

Cytochrome P450 2C19

1 Activities

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Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
AC50	6.7		None, None:None:None