linopirdine
Ligand Summary
Name: linopirdine
PubChem: 3932
Guide to Pharmacology: 2599
ChEMBL: CHEMBL319111
LyCHI: D5LDVLDUNMFY
Target Activities
KCNQ1
Potassium voltage-gated channel subfamily KQT member 1
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 4.4 | |||||
KCNQ2
Potassium voltage-gated channel subfamily KQT member 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.3 | |||||
KCNQ3
Potassium voltage-gated channel subfamily KQT member 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.4 | |||||
KCNQ4
Potassium voltage-gated channel subfamily KQT member 4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 4.9 | |||||
KCNQ5
Potassium voltage-gated channel subfamily KQT member 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 4.8 | |||||
CYP3A4
Cytochrome P450 3A4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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AC50 | 6.3 | None, None:None:None | ||||
CYP2C19
Cytochrome P450 2C19
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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AC50 | 6.7 | None, None:None:None | ||||