SID103904984
Ligand Summary
Target Activities
CDK9
Cyclin-dependent kinase 9
3 Activities
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1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.4 | None, None:None:None | ||||
Ki | 8.4 | None, None:None:None | ||||
IC50 | 8 | J. Med. Chem., (2013) 56:17:6991 | ||||
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.1 | None, None:None:None | ||||
Ki | 9.1 | None, None:None:None | ||||
CSNK1G1
Casein kinase I isoform gamma-1
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
Ki | 7.6 | None, None:None:None | ||||
CSNK1G2
Casein kinase I isoform gamma-2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
Ki | 7.6 | None, None:None:None | ||||
CSNK1D
Casein kinase I isoform delta
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.8 | None, None:None:None | ||||
Ki | 7.8 | None, None:None:None | ||||
GSK3A
Glycogen synthase kinase-3 alpha
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.2 | None, None:None:None | ||||
Ki | 8.2 | None, None:None:None | ||||
JAK2
Tyrosine-protein kinase JAK2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
Ki | 7.7 | None, None:None:None | ||||
CLK4
Dual specificity protein kinase CLK4
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.2 | None, None:None:None | ||||
Ki | 9.2 | None, None:None:None | ||||
STK17A
Serine/threonine-protein kinase 17A
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
Ki | 7.6 | None, None:None:None | ||||
DYRK3
Dual specificity tyrosine-phosphorylation-regulated kinase 3
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8 | None, None:None:None | ||||
Ki | 8 | None, None:None:None | ||||
HIPK2
Homeodomain-interacting protein kinase 2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
Ki | 7.6 | None, None:None:None | ||||
GSK3B
Glycogen synthase kinase-3 beta
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.2 | None, None:None:None | ||||
Ki | 8.2 | None, None:None:None | ||||
CSNK1G3
Casein kinase I isoform gamma-3
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8 | None, None:None:None | ||||
Ki | 8 | None, None:None:None | ||||
DYRK1B
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.2 | None, None:None:None | ||||
Ki | 9.2 | None, None:None:None | ||||
DYRK4
Dual specificity tyrosine-phosphorylation-regulated kinase 4
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8 | None, None:None:None | ||||
Ki | 8 | None, None:None:None | ||||
CDK8
Cyclin-dependent kinase 8
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.8 | None, None:None:None | ||||
Ki | 7.8 | None, None:None:None | ||||
PKN2
Serine/threonine-protein kinase N2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
Ki | 7.7 | None, None:None:None | ||||
CSNK1A1
Casein kinase I isoform alpha
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | None, None:None:None | ||||
Ki | 8.1 | None, None:None:None | ||||
CDC7
Cell division cycle 7-related protein kinase
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.7 | None, None:None:None | ||||
Ki | 9.7 | None, None:None:None | ||||