CHEMBL7463
Ligand Summary
Name: 3-(1-(3-(dimethylamino)propyl)-1H-indol-3-yl)-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione
PubChem: 2396
ChEMBL: CHEMBL7463
LyCHI: CPGXB4PLDPJP
Target Activities
Items per page:
10
1 – 8 of 8
PIM1
Serine/threonine-protein kinase pim-1
3 Activities
PRKCE
Protein kinase C epsilon type
2 Activities
PRKCA
Protein kinase C alpha type
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8 | Bioorg. Med. Chem. Lett., (1995) 5:5:497 | ||||
IC50 | 8.64 | J. Med. Chem., (2009) 52:20:6193 | ||||
PRKCD
Protein kinase C delta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.06 | J. Med. Chem., (2009) 52:20:6193 | ||||
PRKCQ
Protein kinase C theta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.17 | J. Med. Chem., (2009) 52:20:6193 | ||||
PRKCH
Protein kinase C eta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8 | J. Med. Chem., (2009) 52:20:6193 | ||||
PRKCB
Protein kinase C beta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.8 | J. Med. Chem., (2009) 52:20:6193 | ||||
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6 | Eur. J. Med. Chem., (2011) 46:2:618 | ||||