US9260440, 69
Ligand Summary
Target Activities
PARP1
Poly [ADP-ribose] polymerase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.05 | None, (2016) None:None:None | ||||
PARP3
Poly [ADP-ribose] polymerase 3
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.73 | None, (2016) None:None:None | ||||
PARP2
Poly [ADP-ribose] polymerase 2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.3 | None, (2016) None:None:None | ||||
TNKS2
Tankyrase-2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 6.12 | None, (2016) None:None:None | ||||