ivabradine
Ligand Summary
Ivabradine is a pure heart rate lowering agent, acting by selective and specific inhibition of the cardiac pacemaker If current that controls the spontaneous diastolic depolarisation in the sinus node and regulates heart rate. The cardiac effects are specific to the sinus node with no effect on intra-atrial, atrioventricular or intraventricular conduction times, nor on myocardial contractility or ventricular repolarisation.
UNII: 3H48L0LPZQ
PubChem: 132999
Guide to Pharmacology: 2357
ChEMBL: CHEMBL471737
DrugCentral: 3312
LyCHI: 338M8NHVYV2L
Target Activities
9 Activities
Items per page:
10
1 – 9 of 9
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