gallamine
Ligand Summary
A synthetic nondepolarizing blocking drug. The actions of gallamine triethiodide are similar to those of TUBOCURARINE, but this agent blocks the cardiac vagus and may cause sinus tachycardia and, occasionally, hypertension and increased cardiac output. It should be used cautiously in patients at risk from increased heart rate but may be preferred for patients with bradycardia. (From AMA Drug Evaluations Annual, 1992, p198)
UNII: VYJ027LZ05
PubChem: 3450
Guide to Pharmacology: 356
ChEMBL: CHEMBL360055
DrugCentral: 1273
LyCHI: 7GQ3GPZGPVSC
Target Activities
3 Activities
Items per page:
10
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | ||||||
Ki | NEGATIVE ALLOSTERIC MODULATOR | |||||