CHEMBL1236539
Ligand Summary
NCATS Inxight: Drugs: 72271
Name: 7-Hydroxystaurosporine
PubChem: 72271
Guide to Pharmacology: 7907
ChEMBL: CHEMBL1236539
LyCHI: 8NDL1JAFJZTV
Target Activities
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10
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CHEK1
Serine/threonine-protein kinase Chk1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 8.01 | Eur. J. Med. Chem., (2015) 92:None:459 | ||||
PDPK1
3-phosphoinositide-dependent protein kinase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.48000002 | |||||
CHEK2
Serine/threonine-protein kinase Chk2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 5.98000002 | |||||
CDK1
Cyclin-dependent kinase 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.30000019 | |||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 6.30000019 | |||||
LCK
Tyrosine-protein kinase Lck
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.30000019 | |||||
MARK1
Serine/threonine-protein kinase MARK1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.57000017 | |||||
MAPK14
Mitogen-activated protein kinase 14
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.01999998 | |||||
PRKCA
Protein kinase C alpha type
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.53999996 | |||||
PRKCB
Protein kinase C beta type
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.53999996 | |||||