ezetimibe
Ligand Summary
An azetidine derivative and ANTICHOLESTEREMIC AGENT that inhibits intestinal STEROL absorption. It is used to reduce total CHOLESTEROL; LDL CHOLESTEROL, and APOLIPOPROTEINS B in the treatment of HYPERLIPIDEMIAS.
UNII: EOR26LQQ24
PubChem: 150311
Guide to Pharmacology: 6816
ChEMBL: CHEMBL1138
DrugCentral: 1125
LyCHI: B74H5RFQ9SJC
Target Activities
2 Activities
Items per page:
10
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | ||||||
Kd | ANTAGONIST | |||||