aripiprazole
Ligand Summary
A piperazine and quinolone derivative that is used primarily as an antipsychotic agent. It is a partial agonist of SEROTONIN RECEPTOR, 5-HT1A and DOPAMINE D2 RECEPTORS, where it also functions as a post-synaptic antagonist, and an antagonist of SEROTONIN RECEPTOR, 5-HT2A. It is used for the treatment of SCHIZOPHRENIA and BIPOLAR DISORDER, and as an adjunct therapy for the treatment of depression.
UNII: 82VFR53I78
PubChem: 60795
Guide to Pharmacology: 34
ChEMBL: CHEMBL1112
DrugCentral: 242
LyCHI: NY2L457GCS5B
Target Activities
190 Activities
Items per page:
10
1 – 10 of 190
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