Kaempferol
Ligand Summary
Target Activities
CYP1A1
Cytochrome P450 1A1
2 Activities
HSD17B2
Estradiol 17-beta-dehydrogenase 2
2 Activities
CYP1A2
Cytochrome P450 1A2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 7.1 | None, None:None:None | ||||
IC50 | 6.14 | Bioorg. Med. Chem., (2010) 18:17:6310 | ||||
CYP1B1
Cytochrome P450 1B1
2 Activities
CA7
Carbonic anhydrase 7
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | Bioorg. Med. Chem., (2015) 23:22:7219 | ||||
DPP4
Dipeptidyl peptidase 4
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.31 | Eur J Med Chem, (2018) 151:None:145 | ||||
TYR
Tyrosinase
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6 | J. Nat. Prod., (2016) 79:2:281 | ||||
AHR
Aryl hydrocarbon receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.55 | Bioorg. Med. Chem., (2007) 15:15:5047 | ||||
CA12
Carbonic anhydrase 12
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.84 | Bioorg. Med. Chem., (2015) 23:22:7219 | ||||
CYP2C9
Cytochrome P450 2C9
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
AC50 | 8.9 | None, None:None:None | ||||
TRPC5
Short transient receptor potential channel 5
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.41 | J Med Chem, (2019) 62:17:7589 | ||||
CISD1
CDGSH iron-sulfur domain-containing protein 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 6.88 | Bioorg Med Chem Lett, (2016) 26:21:5350 | ||||