CHEMBL4646447
Ligand Summary
Name: N-[4-[(5,11-dimethyl-6-oxo-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]methanesulfonamide
ChEMBL: CHEMBL4646447
LyCHI: BL8RAWYY45QA
Target Activities
DCLK1
Serine/threonine-protein kinase DCLK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.7 | J Med Chem, (2020) 63:14:7817 | ||||