CHEMBL4642915
Ligand Summary
Name: 1-[2-(6-chloro-7-cyclopropyl-thieno[3,2-d]pyrimidin-4-yl)sulfanylacetyl]imidazolidin-4-one
ChEMBL: CHEMBL4642915
LyCHI: AHQTFMXNPSQR
Target Activities
NOTUM
Palmitoleoyl-protein carboxylesterase NOTUM
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.82 | Bioorg Med Chem Lett, (2020) 30:3:126751 | ||||