A-674563
Ligand Summary
Name: A-674563
PubChem: 11314340
Guide to Pharmacology: 5655
ChEMBL: CHEMBL379218
LyCHI: AFFL3QR5PQ81
Target Activities
AKT1
RAC-alpha serine/threonine-protein kinase
4 Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.68 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
PRKG2
cGMP-dependent protein kinase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.72 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
PRKCD
Protein kinase C delta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.57 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
PRKCQ
Protein kinase C theta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.92 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
PRKCE
Protein kinase C epsilon type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.96 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
PRKCH
Protein kinase C eta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.02 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK4
Dual specificity protein kinase CLK4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 9.28 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK1
Dual specificity protein kinase CLK1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.85 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 9.29 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
DYRK1B
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 8.41 | Nat. Biotechnol., (2011) 29:11:1046 | ||||
CIT
Citron Rho-interacting kinase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 7.89 | Nat. Biotechnol., (2011) 29:11:1046 | ||||