Pharos : Ligand Details

Target Activities

AKT1

Tchem

RAC-alpha serine/threonine-protein kinase

4 Activities

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1 – 4 of 4

Activity Type	Activity Value -log(M)	Activity Reference	Publications (PubMed IDs)
IC50	7.85	J. Med. Chem., (2007) 50:13:2990	17523610

Ki	7.96	Bioorg. Med. Chem. Lett., (2006) 16:14:3740	16678413

Kd	7.11999989		22037378

Ki	7.96000004		15956255

PRKG2

Tchem

cGMP-dependent protein kinase 2

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.72		Nat. Biotechnol., (2011) 29:11:1046	22037378

CLK1

Tchem

Dual specificity protein kinase CLK1

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	8.85		Nat. Biotechnol., (2011) 29:11:1046	22037378

PRKCD

Tclin

Protein kinase C delta type

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.57		Nat. Biotechnol., (2011) 29:11:1046	22037378

CIT

Tchem

Citron Rho-interacting kinase

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.89		Nat. Biotechnol., (2011) 29:11:1046	22037378

PRKCQ

Tchem

Protein kinase C theta type

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.92		Nat. Biotechnol., (2011) 29:11:1046	22037378

CLK2

Tchem

Dual specificity protein kinase CLK2

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	9.29		Nat. Biotechnol., (2011) 29:11:1046	22037378

PRKCE

Tchem

Protein kinase C epsilon type

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	7.96		Nat. Biotechnol., (2011) 29:11:1046	22037378

DYRK1B

Tchem

Dual specificity tyrosine-phosphorylation-regulated kinase 1B

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	8.41		Nat. Biotechnol., (2011) 29:11:1046	22037378

PRKCH

Tchem

Protein kinase C eta type

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	8.02		Nat. Biotechnol., (2011) 29:11:1046	22037378

CLK4

Tchem

Dual specificity protein kinase CLK4

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	9.28		Nat. Biotechnol., (2011) 29:11:1046	22037378

DYRK1A

Tchem

Dual specificity tyrosine-phosphorylation-regulated kinase 1A

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	8.68		Nat. Biotechnol., (2011) 29:11:1046	22037378