CHEMBL4569399
Ligand Summary
Name: 1-Isopropyl-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-6-(piperidin-4-yl)-1H-indazole-4-carboxamide
PubChem: 155560721
ChEMBL: CHEMBL4569399
LyCHI: ADYYTZH9JJB2
Target Activities
EZH2
Histone-lysine N-methyltransferase EZH2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.96 | J Med Chem, (2016) 59:16:7617 | ||||
EZH1
Histone-lysine N-methyltransferase EZH1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.21 | J Med Chem, (2016) 59:16:7617 | ||||