CHEMBL4207291
Ligand Summary
Name: N-(1-((5-Cyanopyridin-2-yl)methyl)-1H-pyrazol-3-yl)-2-(3-ethyl-4-(2,2,2-trifluoroethoxy)-phenyl)acetamide
PubChem: 126740608
ChEMBL: CHEMBL4207291
LyCHI: A6KLQTKWNADR
Target Activities
CACNA1H
Voltage-dependent T-type calcium channel subunit alpha-1H
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.11 | J Med Chem, (2017) 60:23:9769 | ||||
CACNA1C
Voltage-dependent L-type calcium channel subunit alpha-1C
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 5.96 | J Med Chem, (2017) 60:23:9769 | ||||
CACNA1G
Voltage-dependent T-type calcium channel subunit alpha-1G
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.96 | J Med Chem, (2017) 60:23:9769 | ||||
CACNA1I
Voltage-dependent T-type calcium channel subunit alpha-1I
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.54 | J Med Chem, (2017) 60:23:9769 | ||||