CHEMBL4476662
Ligand Summary
Name: 2-(4-Chloro-3-methylbenzyl)-5-(4-fluoro-2-methylphenyl)-7-((2-imino-3-methyl-2,3-dihydro-1H-imidazol-1-yl)methyl)-3,4-dihydroisoquinolin-1(2H)-one
PubChem: 153572631
ChEMBL: CHEMBL4476662
LyCHI: A61H4T1MGQTQ
Target Activities
WDR5
WD repeat-containing protein 5
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 10.57 | J Med Chem, (2020) 63:2:656 | ||||