Pharos : Ligand Details - 9P4QCPYWB96C

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: GSK2801

PubChem: 73010930

Guide to Pharmacology: 8233

ChEMBL: CHEMBL3739699

LyCHI: 9P4QCPYWB96C

Target Activities

Explore Associated and Predicted Targets

BAZ2B

Tchem

Bromodomain adjacent to zinc finger domain protein 2B

6 Activities

Items per page:

1 – 6 of 6

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	6.87

Kd	7.22		J. Med. Chem., (2016) 59:4:1410	25799074

Kd	6.87		J. Med. Chem., (2016) 59:4:1410	25799074

Kd	6.85		MedChemComm, (2015) 6:7:1381

IC50	6.44		J. Med. Chem., (2016) 59:7:3087	26982797

IC50	6.37		J. Med. Chem., (2016) 59:4:1410	25799074

BAZ2A

Tchem

Bromodomain adjacent to zinc finger domain protein 2A

4 Activities

Items per page:

1 – 4 of 4

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Kd	6.59

Kd	6.59		J. Med. Chem., (2016) 59:4:1410	25799074

Kd	6.58		MedChemComm, (2015) 6:7:1381

IC50	6.4		J. Med. Chem., (2016) 59:4:1410	25799074