GSK2801
Ligand Summary
Name: GSK2801
PubChem: 73010930
Guide to Pharmacology: 8233
ChEMBL: CHEMBL3739699
LyCHI: 9P4QCPYWB96C
Target Activities
BAZ2B
Bromodomain adjacent to zinc finger domain protein 2B
6 Activities
Items per page:
1 – 6 of 6
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.87 | |||||
Kd | 7.22 | J. Med. Chem., (2016) 59:4:1410 | ||||
Kd | 6.87 | J. Med. Chem., (2016) 59:4:1410 | ||||
Kd | 6.85 | MedChemComm, (2015) 6:7:1381 | ||||
IC50 | 6.44 | J. Med. Chem., (2016) 59:7:3087 | ||||
IC50 | 6.37 | J. Med. Chem., (2016) 59:4:1410 | ||||