CHEMBL3410161
Ligand Summary
Name: (2R,3R)-N1-((S,Z)-1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-phenyl-2-(3,3,3-trifluoropropyl)succinamide
PubChem: 71712019
ChEMBL: CHEMBL3410161
LyCHI: 9L262N5NPGY5
Target Activities
NOTCH1
Neurogenic locus notch homolog protein 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.4 | Bioorg. Med. Chem. Lett., (2015) 25:9:1905 | ||||
NOTCH3
Neurogenic locus notch homolog protein 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.4 | Bioorg. Med. Chem. Lett., (2015) 25:9:1905 | ||||
NOTCH2
Neurogenic locus notch homolog protein 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 9 | Bioorg. Med. Chem. Lett., (2015) 25:9:1905 | ||||
NOTCH4
Neurogenic locus notch homolog protein 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.52 | Bioorg. Med. Chem. Lett., (2015) 25:9:1905 | ||||