GDC-0994
Ligand Summary
Target Activities
MAPK1
Mitogen-activated protein kinase 1
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 9.52 | Bioorg. Med. Chem. Lett., (2015) 25:19:4047 | ||||
Kd | 8.8 | J Med Chem, (2019) 62:24:11004 | ||||
Kd | 8.8 | J Med Chem, (2019) 62:24:11004 | ||||
IC50 | 8.51 | J Med Chem, (2016) 59:12:5650 | ||||
IC50 | 8.48 | None, (2014) None:None:None | ||||
IC50 | 8.48 | None, (2016) None:None:None | ||||
Kd | 7.66 | Science, (2017) 358:6367:None | ||||
MAPK3
Mitogen-activated protein kinase 3
3 Activities
Q6ZSR9
Uncharacterized protein FLJ45252
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Kd | 6.33 | Science, (2017) 358:6367:None | ||||