ALRT 1550
Ligand Summary
Name: ALRT 1550
PubChem: 5287705
Guide to Pharmacology: 2740
ChEMBL: CHEMBL89241
LyCHI: 985232NQJL87
Target Activities
RARB
Retinoic acid receptor beta
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.15 | J. Med. Chem., (1996) 39:14:2659 | ||||
EC50 | 8.66 | J. Med. Chem., (1996) 39:14:2659 | ||||
EC50 | 7.62 | J. Med. Chem., (1996) 39:14:2659 | ||||
Ki | 7.05 | J. Med. Chem., (1996) 39:14:2659 | ||||
RARA
Retinoic acid receptor alpha
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.96 | J. Med. Chem., (1996) 39:14:2659 | ||||
EC50 | 8.4 | J. Med. Chem., (1996) 39:14:2659 | ||||
Ki | 7.2 | J. Med. Chem., (1996) 39:14:2659 | ||||
EC50 | 7.19 | J. Med. Chem., (1996) 39:14:2659 | ||||
RARG
Retinoic acid receptor gamma
3 Activities
RORB
Nuclear receptor ROR-beta
2 Activities
RXRB
Retinoic acid receptor RXR-beta
2 Activities
RXRG
Retinoic acid receptor RXR-gamma
2 Activities
RXRA
Retinoic acid receptor RXR-alpha
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.34 | J. Med. Chem., (1996) 39:14:2659 | ||||