asenapine
Ligand Summary
Name: asenapine
UNII: JKZ19V908O
PubChem: 163091
Guide to Pharmacology: 22
ChEMBL: CHEMBL504548
LyCHI: 96LUGMSY71AA
Target Activities
DRD2
D(2) dopamine receptor
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.92 | |||||
Ki | 8.05 | MedChemComm, (2015) 6:9:1679 | ||||
HTR1B
5-hydroxytryptamine receptor 1B
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
8.1 | ||||||
HTR1D
5-hydroxytryptamine receptor 1D
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
8.4 | ||||||
HTR1E
5-hydroxytryptamine receptor 1E
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
8 | ||||||
HTR2A
5-hydroxytryptamine receptor 2A
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 10.22 | |||||
HRH1
Histamine H1 receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
9.8 | ||||||
DRD3
D(3) dopamine receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.03 | MedChemComm, (2015) 6:9:1679 | ||||
DRD4
D(4) dopamine receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.05 | MedChemComm, (2015) 6:9:1679 | ||||
DRD1
D(1A) dopamine receptor
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 8.05 | MedChemComm, (2015) 6:9:1679 | ||||