CHEMBL4648907
Ligand Summary
Name: N-[2-(2,6-dioxo-3-piperidyl)-1-oxo-isoindolin-4-yl]-2-[[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]pyrimidin-4-yl]amino]acetamide
ChEMBL: CHEMBL4648907
LyCHI: 9466CFQ5XKYW
Target Activities
BRD4
Bromodomain-containing protein 4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.29 | ACS Med Chem Lett, (2020) 11:6:1088 | ||||
CRBN
Protein cereblon
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Ki | 6.89 | ACS Med Chem Lett, (2020) 11:6:1088 | ||||