CHEMBL2147535
Ligand Summary
Name: N-(2-(pyridin-4-yl)pyrido[3,4-d]pyrimidin-4-yl)ethane-1,2-diamine
PubChem: 71452928
ChEMBL: CHEMBL2147535
LyCHI: 8YJ53C9KM25P
Target Activities
LATS1
Serine/threonine-protein kinase LATS1
2 Activities
Items per page:
1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 8.42 | None, None:None:None | ||||
IC50 | 8.42 | |||||
PRKCH
Protein kinase C eta type
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.57 | Bioorg. Med. Chem. Lett., (2011) 21:24:7367 | ||||