CHEMBL451835
Ligand Summary
Name: 4-((5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)ethynyl)benzoic acid
PubChem: 10314719
ChEMBL: CHEMBL451835
LyCHI: 8W7M81MJCU19
Target Activities
RARG
Retinoic acid receptor gamma
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | 9.22 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
RARB
Retinoic acid receptor beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | 9.52 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
RARA
Retinoic acid receptor alpha
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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EC50 | 9.22 | Bioorg. Med. Chem. Lett., (2009) 19:2:489 | ||||
CRABP2
Cellular retinoic acid-binding protein 2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Kd | 6.8 | ACS Med Chem Lett, (2018) 9:12:1297 | ||||