CHEMBL4638458
Ligand Summary
Name: 1-((7-(5-Chloro-2-(((2S,6S)-2,6-dimethylpiperazin-1-yl)methyl)-3-methylphenyl)thieno[3,2-b]pyridin-2-yl)methyl)pyrrolidine-2,5-dione
ChEMBL: CHEMBL4638458
LyCHI: 8TVYVC52HWXB
Target Activities
USP7
Ubiquitin carboxyl-terminal hydrolase 7
2 Activities
KCNH2
Potassium voltage-gated channel subfamily H member 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 5.57 | J Med Chem, (2020) 63:10:5398 | ||||