SID103904190
Ligand Summary
Target Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
Ki | 7.6 | None, None:None:None | ||||
RPS6KA3
Ribosomal protein S6 kinase alpha-3
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.9 | None, None:None:None | ||||
Ki | 7.9 | None, None:None:None | ||||
FLT3
Receptor-type tyrosine-protein kinase FLT3
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.2 | None, None:None:None | ||||
Ki | 8.2 | None, None:None:None | ||||
ROCK1
Rho-associated protein kinase 1
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.9 | None, None:None:None | ||||
Ki | 8.9 | None, None:None:None | ||||
PRKCQ
Protein kinase C theta type
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.1 | None, None:None:None | ||||
Ki | 9.1 | None, None:None:None | ||||
MAP2K1
Dual specificity mitogen-activated protein kinase kinase 1
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
Ki | 7.7 | None, None:None:None | ||||
PRKACA
cAMP-dependent protein kinase catalytic subunit alpha
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | None, None:None:None | ||||
Ki | 8.1 | None, None:None:None | ||||
CLK4
Dual specificity protein kinase CLK4
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9 | None, None:None:None | ||||
Ki | 9 | None, None:None:None | ||||
CLK2
Dual specificity protein kinase CLK2
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.1 | None, None:None:None | ||||
Ki | 8.1 | None, None:None:None | ||||
MELK
Maternal embryonic leucine zipper kinase
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.5 | None, None:None:None | ||||
Ki | 8.5 | None, None:None:None | ||||
DYRK1B
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.8 | None, None:None:None | ||||
Ki | 7.8 | None, None:None:None | ||||
MINK1
Misshapen-like kinase 1
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
Ki | 7.7 | None, None:None:None | ||||
LRRK2
Leucine-rich repeat serine/threonine-protein kinase 2
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.7 | None, None:None:None | ||||
Ki | 8.7 | None, None:None:None | ||||
CDK8
Cyclin-dependent kinase 8
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.3 | None, None:None:None | ||||
Ki | 8.3 | None, None:None:None | ||||
MAP4K4
Mitogen-activated protein kinase kinase kinase kinase 4
2 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
Ki | 7.7 | None, None:None:None | ||||
CSNK1A1
Casein kinase I isoform alpha
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.8 | None, None:None:None | ||||
Ki | 7.8 | None, None:None:None | ||||
CDC7
Cell division cycle 7-related protein kinase
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.5 | None, None:None:None | ||||
Ki | 9.5 | None, None:None:None | ||||
PRKD3
Serine/threonine-protein kinase D3
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.3 | None, None:None:None | ||||
Ki | 8.3 | None, None:None:None | ||||
ROCK2
Rho-associated protein kinase 2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.7 | None, None:None:None | ||||
Ki | 8.7 | None, None:None:None | ||||
CDK5
Cyclin-dependent-like kinase 5
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.5 | None, None:None:None | ||||
Ki | 8.5 | None, None:None:None | ||||
PRKX
cAMP-dependent protein kinase catalytic subunit PRKX
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.5 | None, None:None:None | ||||
Ki | 8.5 | None, None:None:None | ||||