Vorasidenib
Ligand Summary
Target Activities
IDH1
Isocitrate dehydrogenase [NADP] cytoplasmic
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 9.6 | ACS Med Chem Lett, (2020) 11:2:101 | ||||
IDH2
Isocitrate dehydrogenase [NADP], mitochondrial
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 8.15 | ACS Med Chem Lett, (2020) 11:2:101 | ||||