CHEMBL253431
Ligand Summary
Name: (R)-N-(1-(3-(4-cyanophenyl)-4-oxo-3,4-dihydropyrido[2,3-d]pyrimidin-2-yl)ethyl)-N-(2-(ethylsulfonyl)ethyl)-2-(4-fluoro-3-(trifluoromethyl)phenyl)acetamide
PubChem: 16040696
ChEMBL: CHEMBL253431
LyCHI: 87QZB48N84NX
Target Activities
Items per page:
10
1 – 1 of 1
CXCR3
C-X-C chemokine receptor type 3
7 Activities
Items per page:
1 – 7 of 7
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.34 | Bioorg. Med. Chem. Lett., (2012) 22:1:357 | ||||
IC50 | 7.6 | Bioorg. Med. Chem. Lett., (2008) 18:2:688 | ||||
IC50 | 7.6 | Bioorg. Med. Chem. Lett., (2009) 19:17:5200 | ||||
IC50 | 7.96 | Bioorg. Med. Chem. Lett., (2008) 18:2:688 | ||||
IC50 | 7.96 | Bioorg. Med. Chem. Lett., (2009) 19:17:5200 | ||||
IC50 | 7.96 | Bioorg. Med. Chem. Lett., (2009) 19:17:5114 | ||||
IC50 | 7.96 | Bioorg. Med. Chem. Lett., (2012) 22:1:357 | ||||