SID103904462
Ligand Summary
Target Activities
DYRK1A
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.4 | None, None:None:None | ||||
RPS6KA3
Ribosomal protein S6 kinase alpha-3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
DAPK3
Death-associated protein kinase 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
FLT1
Vascular endothelial growth factor receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.2 | None, None:None:None | ||||
PDGFRB
Platelet-derived growth factor receptor beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
FLT3
Receptor-type tyrosine-protein kinase FLT3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
KDR
Vascular endothelial growth factor receptor 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.2 | None, None:None:None | ||||
JAK3
Tyrosine-protein kinase JAK3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
ROCK1
Rho-associated protein kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
MST1R
Macrophage-stimulating protein receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.8 | None, None:None:None | ||||
GSK3A
Glycogen synthase kinase-3 alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.9 | None, None:None:None | ||||
CDK7
Cyclin-dependent kinase 7
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
PRKCQ
Protein kinase C theta type
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
IKBKE
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
PRKACA
cAMP-dependent protein kinase catalytic subunit alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.9 | None, None:None:None | ||||
CLK4
Dual specificity protein kinase CLK4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.5 | None, None:None:None | ||||
CLK2
Dual specificity protein kinase CLK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.1 | None, None:None:None | ||||
GSK3B
Glycogen synthase kinase-3 beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
TYRO3
Tyrosine-protein kinase receptor TYRO3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
MAP4K2
Mitogen-activated protein kinase kinase kinase kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
TBK1
Serine/threonine-protein kinase TBK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
DYRK1B
Dual specificity tyrosine-phosphorylation-regulated kinase 1B
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9 | None, None:None:None | ||||
NTRK3
NT-3 growth factor receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
LRRK2
Leucine-rich repeat serine/threonine-protein kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
MAP4K4
Mitogen-activated protein kinase kinase kinase kinase 4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
PRKAA1
5'-AMP-activated protein kinase catalytic subunit alpha-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
NTRK2
BDNF/NT-3 growth factors receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
PRKD3
Serine/threonine-protein kinase D3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
CDK5
Cyclin-dependent-like kinase 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.2 | None, None:None:None | ||||