CHEMBL4100845
Ligand Summary
Name: 2-(3-([1,1'-biphenyl]-3-yl)-5-cyclopropyl-4-(4-sulfamoylbenzyl)-1H-pyrazol-1-yl)thiazole-4-carboxylic acid
PubChem: 121461710
ChEMBL: CHEMBL4100845
LyCHI: 7ZL28TC5LPMN
Target Activities
LDHA
L-lactate dehydrogenase A chain
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
Kd | 9.48 | J Med Chem, (2017) 60:22:9184 | ||||
IC50 | 7.57 | J Med Chem, (2017) 60:22:9184 | ||||
IC50 | 7.57 | J Med Chem, (2017) 60:22:9184 | ||||
EC50 | 6.6 | J Med Chem, (2017) 60:22:9184 | ||||
LDHB
L-lactate dehydrogenase B chain
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.7 | J Med Chem, (2017) 60:22:9184 | ||||