SID103904402
Ligand Summary
Target Activities
BLK
Tyrosine-protein kinase Blk
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
FLT1
Vascular endothelial growth factor receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
PDGFRB
Platelet-derived growth factor receptor beta
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
FLT4
Vascular endothelial growth factor receptor 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
PDGFRA
Platelet-derived growth factor receptor alpha
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
SRC
Proto-oncogene tyrosine-protein kinase Src
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
KDR
Vascular endothelial growth factor receptor 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
LCK
Tyrosine-protein kinase Lck
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
MST1R
Macrophage-stimulating protein receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
FGFR3
Fibroblast growth factor receptor 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
JAK2
Tyrosine-protein kinase JAK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
LYN
Tyrosine-protein kinase Lyn
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
IRAK1
Interleukin-1 receptor-associated kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
TYK2
Non-receptor tyrosine-protein kinase TYK2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||
FGFR1
Fibroblast growth factor receptor 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
ALK
ALK tyrosine kinase receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
STK17A
Serine/threonine-protein kinase 17A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
TNK2
Activated CDC42 kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
MAP4K5
Mitogen-activated protein kinase kinase kinase kinase 5
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8 | None, None:None:None | ||||
AXL
Tyrosine-protein kinase receptor UFO
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
BTK
Tyrosine-protein kinase BTK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
MAP4K2
Mitogen-activated protein kinase kinase kinase kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
ROS1
Proto-oncogene tyrosine-protein kinase ROS
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
MARK3
MAP/microtubule affinity-regulating kinase 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
LTK
Leukocyte tyrosine kinase receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
BRSK1
Serine/threonine-protein kinase BRSK1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
LRRK2
Leucine-rich repeat serine/threonine-protein kinase 2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9.2 | None, None:None:None | ||||
STK3
Serine/threonine-protein kinase 3
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.9 | None, None:None:None | ||||
LIMK1
LIM domain kinase 1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.8 | None, None:None:None | ||||
PRKAA1
5'-AMP-activated protein kinase catalytic subunit alpha-1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 9 | None, None:None:None | ||||
CHEK2
Serine/threonine-protein kinase Chk2
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.6 | None, None:None:None | ||||
AURKA
Aurora kinase A
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.4 | None, None:None:None | ||||
RET
Proto-oncogene tyrosine-protein kinase receptor Ret
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.9 | None, None:None:None | ||||
ITK
Tyrosine-protein kinase ITK/TSK
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.6 | None, None:None:None | ||||
ERBB4
Receptor tyrosine-protein kinase erbB-4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
PLK4
Serine/threonine-protein kinase PLK4
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.2 | None, None:None:None | ||||