URMC-099
Ligand Summary
Name: URMC-099
PubChem: 54764565
Guide to Pharmacology: 8106
ChEMBL: CHEMBL2436978
LyCHI: 7G137Q8RA7ND
Target Activities
FLT3
Receptor-type tyrosine-protein kinase FLT3
2 Activities
LRRK2
Leucine-rich repeat serine/threonine-protein kinase 2
2 Activities
MAP3K11
Mitogen-activated protein kinase kinase kinase 11
2 Activities
MAP3K9
Mitogen-activated protein kinase kinase kinase 9
2 Activities
ABL1
Tyrosine-protein kinase ABL1
2 Activities
DLK1
Protein delta homolog 1
2 Activities
DAPK3
Death-associated protein kinase 3
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.82 | |||||
MAP3K10
Mitogen-activated protein kinase kinase kinase 10
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 7.38 | |||||
MAP3K2
Mitogen-activated protein kinase kinase kinase 2
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.18 | |||||