Pharos : Ligand Details - 7CLT73A6ZVBQ

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Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: tamibarotene

PubChem: 108143

Guide to Pharmacology: 2648

ChEMBL: CHEMBL25202

LyCHI: 7CLT73A6ZVBQ

Target Activities

Explore Associated and Predicted Targets

RARA

Tclin

Retinoic acid receptor alpha

5 Activities

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1 – 5 of 5

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
-	6.9			3184125 7791761 10637371

EC50	7.35			20925433

Ki	8.19		J. Med. Chem., (1997) 40:26:4222	9435893

EC50	7.35		J. Med. Chem., (2010) 53:19:6779	20925433

IC50	7.11		J. Med. Chem., (2000) 43:3:409	10669568

RARB

Tclin

Retinoic acid receptor beta

2 Activities

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1 – 2 of 2

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.63			20925433

Ki	7.52		J. Med. Chem., (1997) 40:26:4222	9435893

RARG

Tclin

Retinoic acid receptor gamma

1 Activities

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1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
EC50	6.23			20925433