Pharos : Ligand Details - 6Y262D6APNP7

You are using an outdated browser. Please upgrade your browser to improve your experience.

Ligand Summary

Ligand Structure

Rendered image for the query structure

Synonyms & Links

Name: 9a,11a-Dimethyl-7-oxo-2,3,3a,3b,4,5,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-cyclopenta[i]phenanthridine-1-carboxylic acid methyl ester

PubChem: 10065301

ChEMBL: CHEMBL297524

LyCHI: 6Y262D6APNP7

Target Activities

SRD5A1

Tclin

3-oxo-5-alpha-steroid 4-dehydrogenase 1

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	6.82		J. Med. Chem., (1993) 36:26:4313	8277514

Ki	6.82		J. Med. Chem., (1997) 40:9:1293	9135028

Ki	6.82		J. Med. Chem., (1994) 37:15:2352	8057283

SRD5A2

Tclin

3-oxo-5-alpha-steroid 4-dehydrogenase 2

3 Activities

Items per page:

1 – 3 of 3

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
IC50	8.49		J. Med. Chem., (1993) 36:26:4313	8277514

IC50	8.49		J. Med. Chem., (1997) 40:9:1293	9135028

IC50	8.49		J. Med. Chem., (1994) 37:15:2352	8057283

HSD3B1

Tchem

3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1

1 Activities

Items per page:

1 – 1 of 1

Activity Type	Activity Value -log(M)	Mechanism of Action	Activity Reference	Publications (PubMed IDs)
Ki	7.92		J. Med. Chem., (1997) 40:9:1293	9135028