FTY720-P(R)
Ligand Summary
Target Activities
S1PR1
Sphingosine 1-phosphate receptor 1
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 9.85 | Bioorg. Med. Chem. Lett., (2010) 20:5:1485 | ||||
IC50 | 9.8 | Bioorg. Med. Chem. Lett., (2010) 20:5:1485 | ||||
EC50 | 9.17 | Bioorg. Med. Chem. Lett., (2007) 17:2:491 | ||||
EC50 | 7.66 | J. Med. Chem., (2005) 48:16:5373 | ||||
EC50 | 7.63 | Bioorg. Med. Chem. Lett., (2010) 20:7:2264 | ||||
S1PR3
Sphingosine 1-phosphate receptor 3
4 Activities
Items per page:
1 – 4 of 4
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 8.77 | Bioorg. Med. Chem. Lett., (2007) 17:2:491 | ||||
EC50 | 8.6 | Bioorg. Med. Chem. Lett., (2010) 20:5:1485 | ||||
EC50 | 7.79 | Bioorg. Med. Chem. Lett., (2010) 20:7:2264 | ||||
EC50 | 7.54 | J. Med. Chem., (2005) 48:16:5373 | ||||
S1PR4
Sphingosine 1-phosphate receptor 4
3 Activities
Items per page:
1 – 3 of 3
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
EC50 | 9.15 | Bioorg. Med. Chem. Lett., (2010) 20:5:1485 | ||||
EC50 | 7.73 | Bioorg. Med. Chem. Lett., (2007) 17:2:491 | ||||
EC50 | 7.1 | J. Med. Chem., (2005) 48:16:5373 | ||||