CHEMBL4544978
Ligand Summary
Name: N-((4-Ethyl-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-isopropyl-6-(6-(4-isopropylpiperazin-1-yl)pyridin-3-yl)-1H-indazole-4-carboxamide
PubChem: 155552788
ChEMBL: CHEMBL4544978
LyCHI: 6KRM5H93XZCF
Target Activities
EZH2
Histone-lysine N-methyltransferase EZH2
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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IC50 | 7.92 | J Med Chem, (2016) 59:16:7617 | ||||
EZH1
Histone-lysine N-methyltransferase EZH1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
IC50 | 6.09 | J Med Chem, (2016) 59:16:7617 | ||||