CHEMBL4172856
Ligand Summary
Name: 1-Methylcyclopropyl 4-(3-((3-((3,5-bis(trifluoromethyl)benzyl)(methyl)carbamoyl)-1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)oxy)propyl)piperidine-1-carboxylate
PubChem: 137628633
ChEMBL: CHEMBL4172856
LyCHI: 6DY1UYS8QJNB
Target Activities
SGMS2
Phosphatidylcholine:ceramide cholinephosphotransferase 2
5 Activities
Items per page:
1 – 5 of 5
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 8.19 | Eur J Med Chem, (2017) 136:None:283 | ||||
Kd | 7.55 | Eur J Med Chem, (2017) 136:None:283 | ||||
Kd | 7.52 | Eur J Med Chem, (2017) 136:None:283 | ||||
Kd | 7.42 | Eur J Med Chem, (2017) 136:None:283 | ||||
Kd | 6.62 | Eur J Med Chem, (2017) 136:None:283 | ||||
SGMS1
Phosphatidylcholine:ceramide cholinephosphotransferase 1
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6 | Eur J Med Chem, (2017) 136:None:283 | ||||