CHEMBL3938615
Ligand Summary
Name: 1-(4-{[(2S,4R)-2-(2,4-dichlorophenyl)-2-(imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy}phenyl)-4-trifluoromethanesulfonylpiperazine
PubChem: 77846787
ChEMBL: CHEMBL3938615
LyCHI: 5P9UDFB1KDC8
Target Activities
CYP3A4
Cytochrome P450 3A4
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.47 | Bioorg Med Chem Lett, (2016) 26:23:5825 | ||||
CYP19A1
Aromatase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 6.1 | Bioorg Med Chem Lett, (2016) 26:23:5825 | ||||
CYP17A1
Steroid 17-alpha-hydroxylase/17,20 lyase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.17 | Bioorg Med Chem Lett, (2016) 26:23:5825 | ||||
CYP11B1
Cytochrome P450 11B1, mitochondrial
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.5 | Bioorg Med Chem Lett, (2016) 26:23:5825 | ||||
CYP21A2
Steroid 21-hydroxylase
1 Activities
Items per page:
1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
|---|---|---|---|---|---|---|
IC50 | 7.31 | Bioorg Med Chem Lett, (2016) 26:23:5825 | ||||