SID103904315
Ligand Summary
Target Activities
KDR
Vascular endothelial growth factor receptor 2
2 Activities
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1 – 2 of 2
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.4 | None, None:None:None | ||||
IC50 | 7.82 | Bioorg. Med. Chem. Lett., (2012) 22:9:3208 | ||||
BLK
Tyrosine-protein kinase Blk
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.9 | None, None:None:None | ||||
FYN
Tyrosine-protein kinase Fyn
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 7.7 | None, None:None:None | ||||
CSF1R
Macrophage colony-stimulating factor 1 receptor
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.5 | None, None:None:None | ||||
ABL1
Tyrosine-protein kinase ABL1
1 Activities
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Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.9 | None, None:None:None | ||||
FLT1
Vascular endothelial growth factor receptor 1
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 9.4 | None, None:None:None | ||||
KIT
Mast/stem cell growth factor receptor Kit
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.3 | None, None:None:None | ||||
LYN
Tyrosine-protein kinase Lyn
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
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Ki | 8.1 | None, None:None:None | ||||
MET
Hepatocyte growth factor receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
FER
Tyrosine-protein kinase Fer
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
FRK
Tyrosine-protein kinase FRK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
AXL
Tyrosine-protein kinase receptor UFO
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.7 | None, None:None:None | ||||
BTK
Tyrosine-protein kinase BTK
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 7.6 | None, None:None:None | ||||
NTRK3
NT-3 growth factor receptor
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.5 | None, None:None:None | ||||
AURKA
Aurora kinase A
1 Activities
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1 – 1 of 1
Activity Type | Activity Value -log(M) | Mechanism of Action | Activity Reference | Publications (PubMed IDs) | ||
---|---|---|---|---|---|---|
Ki | 8.2 | None, None:None:None | ||||